Novel synthesis of arylethynyl heterocyles

Author

Soley, Roger

Albericio Palomera, Fernando

Álvarez Domingo, Mercedes

Publication date

2014-07-04T09:46:49Z

2014-07-04T09:46:49Z

2007-05-02

2014-07-04T09:46:51Z

Abstract

A new and easy synthesis of 2-arylethynyl-indole and 2-arylethynyl-pyrrole is described. N-deprotection and subsequent base-catalyzed elimination of N-tosylheteroaryl benzyl ketones are the key steps of the process.

Document Type

Article
Accepted version

Language

English

Subjects and keywords

Síntesi orgànica; Compostos heterocíclics; Acetilè; Organic synthesis; Heterocyclic compounds; Acetylene

Publisher

Georg Thieme Verlag

Related items

Versió postprint del document publicat a: http://dx.doi.org/10.1055/s-2007-966041

Synthesis. Journal of Synthetic Organic Chemistry, 2007, num. 10, p. 1559-1565

http://dx.doi.org/10.1055/s-2007-966041

Rights

(c) Georg Thieme Verlag, 2007